Simple exploration of 14452-30-3

According to the analysis of related databases, 14452-30-3, the application of this compound in the production field has become more and more popular.

Each compound has different characteristics, and only by selecting the characteristics of the compound suitable for a specific situation can the compound be applied on a large scale. 14452-30-3, name is 1-(3-Iodophenyl)ethanone, This compound has unique chemical properties. The synthetic route is as follows., Recommanded Product: 1-(3-Iodophenyl)ethanone

1-[3-(2,6-difluorobenzyl)-phenyl]-ethanone (8A). A suspension of Dibromoethane (0.28 mL, 0.0032 mole) in 35 mL of THF under Argon was treated with activated zinc (10.5 g, 0.161 mole) and heated to reflux 2 times for 30 seconds each time. The suspension was then cooled in a salt water ice bath to -8 C. and 2,6-Difluorobenzyl bromide (16.8 g, 0.081 mole) in 20 mL of THF was added dropwise. After addition was completed the reaction was allowed to stir at 0 C., for 1 hour. In a separate flask was added Bis(dibenzylideneacetone)palladium (3.1 g, 0.00537 mole), Tri(2-furyl) phosphine (2.5 g, 0.0107 mole), and 3-iodoacetophenone (13 g, 0.0537 mole) to 40 mL of THF and cooled to 0 C. The zinc suspension was then cannulated into the 3-iodoacetophenone mixture and the ice bath was removed. After 18 hours the mixture was filtered through a pad of celite and washed several times with EtOAc and then the solvents were removed under reduced pressure. The residue was treated with 150 mL of a saturated aqueous solution of NH4Cl and extracted with EtOAc three times, the combined organic layers were dried over NaSO4, filtered and evaporated to give a brown oil. This crude product was flash chromatographed with 15% EtOAc/Hexanes to give 1-[3-(2,6-difluoro-benzyl)-phenyl]-ethanone (8A) as a yellow oil. Rf=0.56 (15% EtOAc/Hexanes). 1H NMR (400 MHz, CDCl3) delta 7.86 (s, 1H), 7.78 (d, j=7.6 Hz, 1H), 7.45 (d, j=8.3 Hz, 1H), 7.36 (t, j=7.6 Hz 1H), 7.19 (m, 1H), 6.89 (m, 2H), 4.07 (s, 2H), 2.57 (s, 3H)

According to the analysis of related databases, 14452-30-3, the application of this compound in the production field has become more and more popular.

Reference:
Patent; Payne, Linda S.; Tran, Lekhanh O.; Zhuang, Linghang H.; Young, Steven D.; Egbertson, Melissa S.; Wai, John S.; Embrey, Mark W.; Fisher, Thorsten E.; Guare, James P.; Langford, H. Marie; Melamed, Jeffrey Y.; Clark, David L.; US2003/229079; (2003); A1;,
Iodide – Wikipedia,
Iodide – an overview | ScienceDirect Topics – ScienceDirect.com